{"doi":"10.17615/wa7e-m156","title":"UNC2025, a MERTK Small-Molecule Inhibitor, Is Therapeutically Effective Alone and in Combination with Methotrexate in Leukemia Models","abstract":"MERTK tyrosine kinase is ectopically expressed in 30–50% of acute lymphoblastic leukemias (ALL) and over 80% of acute myeloid leukemias (AML) and is a potential therapeutic target. Here, we evaluated the utility of UNC2025, a MERTK tyrosine kinase inhibitor, for treatment of acute leukemia.","journal":"UNC Libraries","year":2020,"id":141100,"datarank":0.0,"base_score":0.0,"endowment":0.0,"self_citation_contribution":0.0,"citation_network_contribution":0.0,"self_endowment_contribution":0.0,"citer_contribution":0.0,"corpus_percentile":null,"corpus_rank":null,"citation_count":0,"citer_count":0,"citers_with_citation_signal":0,"citers_with_endowment":0,"datacite_reuse_total":0,"is_dataset":false,"is_dataset_confidence":0.9523,"is_data_producer":false,"deposit_databanks":null,"is_oa":true,"file_count":0,"downloads":0,"has_version_chain":false,"published_date":"2020-01-01","fair_score":null,"fair_percentile":null,"algorithm_id":"datarank_citation_only_1hop_v6","ranking_scope":"data_only","authors":[{"id":278820,"name":"Jeffrey Tyner","orcid":"0000-0002-2133-0960","position":1,"is_corresponding":false},{"id":606013,"name":"Lauren S. Page","orcid":null,"position":2,"is_corresponding":false},{"id":472949,"name":"Alisa B. Lee‐Sherick","orcid":"0000-0002-1177-7208","position":3,"is_corresponding":false},{"id":275365,"name":"Douglas K. Graham","orcid":"0000-0002-6201-6900","position":4,"is_corresponding":false},{"id":605897,"name":"Madeline G. Huey","orcid":"0000-0002-7456-9537","position":5,"is_corresponding":false},{"id":606640,"name":"Kristen M. Jacobsen","orcid":null,"position":6,"is_corresponding":false},{"id":594025,"name":"H Shelton Earp","orcid":null,"position":7,"is_corresponding":false},{"id":605501,"name":"Amanda A. Hill","orcid":"0009-0009-9392-1717","position":8,"is_corresponding":false},{"id":606014,"name":"Gregory Kirkpatrick","orcid":null,"position":9,"is_corresponding":false},{"id":392226,"name":"Stephen V. Frye","orcid":"0000-0002-2415-2215","position":10,"is_corresponding":false},{"id":606641,"name":"Fatma Eryildiz","orcid":null,"position":11,"is_corresponding":false},{"id":105115,"name":"Stephanie A. Montgomery","orcid":"0000-0001-8012-5302","position":12,"is_corresponding":false},{"id":392225,"name":"Xiaodong Wang","orcid":"0000-0003-3293-7538","position":13,"is_corresponding":false},{"id":275364,"name":"Deborah DeRyckere","orcid":"0000-0002-7457-9006","position":14,"is_corresponding":false},{"id":515169,"name":"Weihe Zhang","orcid":"0000-0003-2923-9130","position":0,"is_corresponding":true}],"reference_count":0,"raw_metadata":null,"created_at":"2026-07-18T23:17:20.701143Z","pmid":null,"pmcid":null,"fwci":null,"citation_percentile":null,"influential_citations":0,"oa_status":null,"license":null,"views":0,"total_file_size_bytes":0,"version_count":0,"fair_f":null,"fair_a":null,"fair_i":null,"fair_r":null,"fair_zscore":null,"fair_rationale":null,"fair_model":null,"fair_agent_version":null,"fair_fulltext_source":null,"fair_has_llm":null,"fair_computed_at":null,"clinical_trials":[],"software_tools":[],"db_accessions":[],"linked_datasets":[],"topics":[]}