{"doi":"10.1128/aac.00684-23","title":"Tartrolon E, a secondary metabolite of a marine symbiotic bacterium, is a potent inhibitor of asexual and sexual <i>Plasmodium falciparum</i>","abstract":"ABSTRACT Due to the spread of resistance to front-line artemisinin derivatives worldwide, there is a need for new antimalarials. Tartrolon E (TrtE), a secondary metabolite of a symbiotic bacterium of marine bivalve mollusks, is a promising antimalarial because it inhibits the growth of sexual and asexual blood stages of Plasmodium falciparum at sub-nanomolar levels. The potency of TrtE warrants further investigation into its mechanism of action, cytotoxicity, and ease with which parasites may evolve resistance to it.","journal":"Antimicrobial Agents and Chemotherapy","year":2024,"id":448205,"datarank":0.0,"base_score":0.0,"endowment":0.0,"self_citation_contribution":0.0,"citation_network_contribution":0.0,"self_endowment_contribution":0.0,"citer_contribution":0.0,"corpus_percentile":null,"corpus_rank":null,"citation_count":5,"citer_count":0,"citers_with_citation_signal":0,"citers_with_endowment":0,"datacite_reuse_total":0,"is_dataset":false,"is_dataset_confidence":0.9562,"is_data_producer":false,"deposit_databanks":null,"is_oa":true,"file_count":0,"downloads":0,"has_version_chain":false,"published_date":"2024-01-01","fair_score":null,"fair_percentile":null,"algorithm_id":"datarank_citation_only_1hop_v6","ranking_scope":"data_only","authors":[{"id":748079,"name":"Rapatbhorn Patrapuvich","orcid":"0000-0001-8214-5710","position":1,"is_corresponding":false},{"id":748896,"name":"Devaraja G. Mudeppa","orcid":null,"position":2,"is_corresponding":false},{"id":472396,"name":"Sreekanth Kokkonda","orcid":null,"position":3,"is_corresponding":false},{"id":982149,"name":"Rimi Chakrabarti","orcid":"0000-0002-0336-7428","position":4,"is_corresponding":false},{"id":360642,"name":"Patchara Sriwichai","orcid":"0000-0003-2065-0660","position":5,"is_corresponding":false},{"id":445336,"name":"Roberta M. O’Connor","orcid":"0000-0003-2757-754X","position":6,"is_corresponding":false},{"id":471522,"name":"Pradipsinh K. Rathod","orcid":"0000-0001-7394-1360","position":7,"is_corresponding":false},{"id":433759,"name":"John White","orcid":"0000-0001-7895-4443","position":8,"is_corresponding":false},{"id":982695,"name":"Laura Chery-Karschney","orcid":null,"position":0,"is_corresponding":true}],"reference_count":18,"raw_metadata":null,"created_at":"2026-07-19T02:02:08.018689Z","pmid":"38193705","pmcid":null,"fwci":null,"citation_percentile":null,"influential_citations":0,"oa_status":null,"license":null,"views":0,"total_file_size_bytes":0,"version_count":0,"fair_f":null,"fair_a":null,"fair_i":null,"fair_r":null,"fair_zscore":null,"fair_rationale":null,"fair_model":null,"fair_agent_version":null,"fair_fulltext_source":null,"fair_has_llm":null,"fair_computed_at":null,"clinical_trials":[],"software_tools":[],"db_accessions":[],"linked_datasets":[],"topics":[]}