{"doi":"10.1039/d4cb00206g","title":"Biochemical characterization and discovery of inhibitors for <i>Pf</i> Sir2A: new tricks for an old enzyme","abstract":"Pf Sir2A controls the var virulence gene expression in malaria parasites. Inhibitors targeting Pf Sir2A are potential antimalarial agents. In the current study, 3-TYP and NR are identified as lead compounds for further inhibitor development.","journal":"RSC Chemical Biology","year":2025,"id":560697,"datarank":0.0,"base_score":0.0,"endowment":0.0,"self_citation_contribution":0.0,"citation_network_contribution":0.0,"self_endowment_contribution":0.0,"citer_contribution":0.0,"corpus_percentile":null,"corpus_rank":null,"citation_count":0,"citer_count":0,"citers_with_citation_signal":0,"citers_with_endowment":0,"datacite_reuse_total":0,"is_dataset":false,"is_dataset_confidence":0.9552,"is_data_producer":false,"deposit_databanks":null,"is_oa":true,"file_count":0,"downloads":0,"has_version_chain":false,"published_date":"2025-01-01","fair_score":null,"fair_percentile":null,"algorithm_id":"datarank_citation_only_1hop_v6","ranking_scope":"data_only","authors":[{"id":1354143,"name":"Emily Boyle","orcid":"0000-0001-8803-3939","position":1,"is_corresponding":false},{"id":452929,"name":"Alyson M. Curry","orcid":"0000-0003-2996-4519","position":2,"is_corresponding":false},{"id":406422,"name":"Yana Cen","orcid":"0000-0001-6436-5744","position":3,"is_corresponding":false},{"id":441367,"name":"Dickson Donu","orcid":"0000-0002-5686-2609","position":0,"is_corresponding":true}],"reference_count":49,"raw_metadata":null,"created_at":"2026-07-19T02:55:46.921885Z","pmid":"39897407","pmcid":null,"fwci":null,"citation_percentile":null,"influential_citations":0,"oa_status":null,"license":null,"views":0,"total_file_size_bytes":0,"version_count":0,"fair_f":null,"fair_a":null,"fair_i":null,"fair_r":null,"fair_zscore":null,"fair_rationale":null,"fair_model":null,"fair_agent_version":null,"fair_fulltext_source":null,"fair_has_llm":null,"fair_computed_at":null,"clinical_trials":[],"software_tools":[],"db_accessions":[],"linked_datasets":[],"topics":[]}