{"doi":"10.1039/d3md00058c","title":"<i>Mycobacterium tuberculosis</i> CitA activity is modulated by cysteine oxidation and pyruvate binding","abstract":"values of 6.6 and 10.9 μM. A crystal structure of CitA modified by Ebselen was solved, but significant structural changes were lacking. Considering that covalent modification of C143 inactivates CitA and the proximity of C143 to the pyruvate binding site, this suggests that structural and/or chemical changes in this sub-domain are responsible for regulating CitA enzymatic activity.","journal":"RSC Medicinal Chemistry","year":2023,"id":376743,"datarank":0.0,"base_score":0.0,"endowment":0.0,"self_citation_contribution":0.0,"citation_network_contribution":0.0,"self_endowment_contribution":0.0,"citer_contribution":0.0,"corpus_percentile":null,"corpus_rank":null,"citation_count":3,"citer_count":0,"citers_with_citation_signal":0,"citers_with_endowment":0,"datacite_reuse_total":0,"is_dataset":false,"is_dataset_confidence":0.9547,"is_data_producer":false,"deposit_databanks":null,"is_oa":true,"file_count":0,"downloads":0,"has_version_chain":false,"published_date":"2023-01-01","fair_score":null,"fair_percentile":null,"algorithm_id":"datarank_citation_only_1hop_v6","ranking_scope":"data_only","authors":[{"id":1136214,"name":"Lorenza Favrot","orcid":null,"position":1,"is_corresponding":false},{"id":1139922,"name":"Cécile Petit","orcid":"0000-0002-1864-6630","position":2,"is_corresponding":false},{"id":849077,"name":"Melvin Yamsek","orcid":null,"position":3,"is_corresponding":false},{"id":685394,"name":"Sarbjit Singh","orcid":"0000-0001-5719-967X","position":4,"is_corresponding":false},{"id":658274,"name":"Jayapal Reddy Mallareddy","orcid":"0000-0003-0440-6617","position":5,"is_corresponding":false},{"id":415308,"name":"Sandeep Rana","orcid":"0000-0001-5802-5970","position":6,"is_corresponding":false},{"id":415310,"name":"Amarnath Natarajan","orcid":"0000-0001-5067-0203","position":7,"is_corresponding":false},{"id":431733,"name":"Donald R. Ronning","orcid":"0000-0003-2583-8849","position":8,"is_corresponding":false},{"id":1139921,"name":"Rasangi Pathirage","orcid":"0000-0002-8751-8042","position":0,"is_corresponding":true}],"reference_count":54,"raw_metadata":null,"created_at":"2026-07-19T01:16:32.368674Z","pmid":"37252106","pmcid":null,"fwci":null,"citation_percentile":null,"influential_citations":0,"oa_status":null,"license":null,"views":0,"total_file_size_bytes":0,"version_count":0,"fair_f":null,"fair_a":null,"fair_i":null,"fair_r":null,"fair_zscore":null,"fair_rationale":null,"fair_model":null,"fair_agent_version":null,"fair_fulltext_source":null,"fair_has_llm":null,"fair_computed_at":null,"clinical_trials":[],"software_tools":[],"db_accessions":[],"linked_datasets":[],"topics":[]}