{"doi":"10.1039/d3cb00103b","title":"Development of a covalent cereblon-based PROTAC employing a fluorosulfate warhead","abstract":", and in cells the BRD4 degrader is insensitive to wash-out and competition by potent reversible CRBN ligands, reflecting enhanced pharmacodynamics. We anticipate that covalent CRBN-based PROTACs will enhance degradation efficiencies, thus expanding the scope of addressable targets using the heterobifunctional degrader modality.","journal":"RSC Chemical Biology","year":2023,"id":321992,"datarank":0.0,"base_score":0.0,"endowment":0.0,"self_citation_contribution":0.0,"citation_network_contribution":0.0,"self_endowment_contribution":0.0,"citer_contribution":0.0,"corpus_percentile":null,"corpus_rank":null,"citation_count":42,"citer_count":0,"citers_with_citation_signal":0,"citers_with_endowment":0,"datacite_reuse_total":0,"is_dataset":false,"is_dataset_confidence":0.9636,"is_data_producer":false,"deposit_databanks":null,"is_oa":true,"file_count":0,"downloads":0,"has_version_chain":false,"published_date":"2023-01-01","fair_score":null,"fair_percentile":null,"algorithm_id":"datarank_citation_only_1hop_v6","ranking_scope":"data_only","authors":[{"id":1034890,"name":"Leah Ragosta","orcid":"0009-0007-9977-942X","position":1,"is_corresponding":false},{"id":855933,"name":"Fidel Huerta","orcid":"0000-0002-6721-6506","position":2,"is_corresponding":false},{"id":855934,"name":"Hu Liu","orcid":"0000-0002-5237-6419","position":3,"is_corresponding":false},{"id":227599,"name":"Scott B. Ficarro","orcid":"0000-0002-1521-7996","position":4,"is_corresponding":false},{"id":856802,"name":"Justin T. Cruite","orcid":null,"position":5,"is_corresponding":false},{"id":855935,"name":"Rebecca J. Metivier","orcid":"0000-0001-9929-6857","position":6,"is_corresponding":false},{"id":299772,"name":"Katherine A. Donovan","orcid":"0000-0002-8539-5106","position":7,"is_corresponding":false},{"id":227615,"name":"Jarrod A. Marto","orcid":"0000-0003-2086-1134","position":8,"is_corresponding":false},{"id":262829,"name":"Eric S. Fischer","orcid":"0000-0001-7337-6306","position":9,"is_corresponding":false},{"id":588890,"name":"Breanna L. Zerfas","orcid":"0000-0002-5242-0547","position":10,"is_corresponding":false},{"id":655802,"name":"Lyn H. Jones","orcid":"0000-0002-8388-5865","position":11,"is_corresponding":false},{"id":262828,"name":"Radosław P. Nowak","orcid":"0000-0002-0605-0071","position":0,"is_corresponding":true}],"reference_count":42,"raw_metadata":null,"created_at":"2026-07-19T01:07:37.596550Z","pmid":"37920397","pmcid":null,"fwci":null,"citation_percentile":null,"influential_citations":0,"oa_status":null,"license":null,"views":0,"total_file_size_bytes":0,"version_count":0,"fair_f":null,"fair_a":null,"fair_i":null,"fair_r":null,"fair_zscore":null,"fair_rationale":null,"fair_model":null,"fair_agent_version":null,"fair_fulltext_source":null,"fair_has_llm":null,"fair_computed_at":null,"clinical_trials":[],"software_tools":[],"db_accessions":[],"linked_datasets":[],"topics":[]}