{"doi":"10.1039/d0md00382d","title":"Selective degradation-inducing probes for studying cereblon (CRBN) biology","abstract":"Thorough compound characterization by combination western and proteomic analysis identified ZXH-4-130 and ZXH-4-137 as potent and selective small molecule degraders of cereblon (CRBN).","journal":"RSC Medicinal Chemistry","year":2021,"id":170986,"datarank":0.0,"base_score":0.0,"endowment":0.0,"self_citation_contribution":0.0,"citation_network_contribution":0.0,"self_endowment_contribution":0.0,"citer_contribution":0.0,"corpus_percentile":null,"corpus_rank":null,"citation_count":27,"citer_count":0,"citers_with_citation_signal":0,"citers_with_endowment":0,"datacite_reuse_total":0,"is_dataset":false,"is_dataset_confidence":0.9622,"is_data_producer":false,"deposit_databanks":null,"is_oa":true,"file_count":0,"downloads":0,"has_version_chain":false,"published_date":"2021-01-01","fair_score":null,"fair_percentile":null,"algorithm_id":"datarank_citation_only_1hop_v6","ranking_scope":"data_only","authors":[{"id":228754,"name":"Guangyan Du","orcid":"0000-0002-6413-8741","position":1,"is_corresponding":false},{"id":463161,"name":"Jonathan W. Bushman","orcid":"0000-0002-8230-6315","position":2,"is_corresponding":false},{"id":228753,"name":"Zhixiang He","orcid":"0000-0002-4493-0336","position":3,"is_corresponding":false},{"id":226576,"name":"Tinghu Zhang","orcid":"0000-0003-1028-8020","position":4,"is_corresponding":false},{"id":262829,"name":"Eric S. Fischer","orcid":"0000-0001-7337-6306","position":5,"is_corresponding":false},{"id":226581,"name":"Nathanael S. Gray","orcid":"0000-0001-5354-7403","position":6,"is_corresponding":false},{"id":704714,"name":"Chelsea E. Powell","orcid":"0000-0001-7624-1116","position":0,"is_corresponding":true}],"reference_count":46,"raw_metadata":null,"created_at":"2026-07-18T23:46:28.747384Z","pmid":"34458741","pmcid":null,"fwci":null,"citation_percentile":null,"influential_citations":0,"oa_status":null,"license":null,"views":0,"total_file_size_bytes":0,"version_count":0,"fair_f":null,"fair_a":null,"fair_i":null,"fair_r":null,"fair_zscore":null,"fair_rationale":null,"fair_model":null,"fair_agent_version":null,"fair_fulltext_source":null,"fair_has_llm":null,"fair_computed_at":null,"clinical_trials":[],"software_tools":[],"db_accessions":[],"linked_datasets":[],"topics":[]}