{"doi":"10.1021/acsmedchemlett.7b00476","title":"From RORγt Agonist to Two Types of RORγt Inverse Agonists","abstract":null,"journal":"ACS Medicinal Chemistry Letters","year":2018,"id":14271,"datarank":1.1834071056028295,"base_score":3.4339872044851463,"endowment":3.4339872044851463,"self_citation_contribution":0.515098080672772,"citation_network_contribution":0.6683090249300576,"self_endowment_contribution":0.515098080672772,"citer_contribution":0.6683090249300576,"corpus_percentile":null,"corpus_rank":null,"citation_count":30,"citer_count":21,"citers_with_citation_signal":20,"citers_with_endowment":20,"datacite_reuse_total":0,"is_dataset":false,"is_dataset_confidence":null,"is_oa":false,"file_count":0,"downloads":0,"has_version_chain":false,"published_date":null,"fair_score":null,"fair_percentile":null,"algorithm_id":"datarank_citation_only_1hop_v6","ranking_scope":"data_only","authors":[{"id":113512,"name":"Wei Cai","orcid":null,"position":1,"is_corresponding":false},{"id":113513,"name":"Ting Tang","orcid":null,"position":2,"is_corresponding":false},{"id":113514,"name":"Qian Liu","orcid":null,"position":3,"is_corresponding":false},{"id":17728,"name":"Ting Yang","orcid":"0000-0001-8872-8749","position":4,"is_corresponding":false},{"id":113515,"name":"Liuqing Yang","orcid":"0000-0002-0086-2909","position":5,"is_corresponding":false},{"id":113516,"name":"Yingli Ma","orcid":null,"position":6,"is_corresponding":false},{"id":96887,"name":"Guifeng Zhang","orcid":"0000-0002-7885-4968","position":7,"is_corresponding":false},{"id":113517,"name":"Yafei Huang","orcid":null,"position":8,"is_corresponding":false},{"id":113518,"name":"Xiaoxia Song","orcid":null,"position":9,"is_corresponding":false},{"id":113519,"name":"Lisa A. Orband-Miller","orcid":null,"position":10,"is_corresponding":false},{"id":113520,"name":"Qianqian Wu","orcid":null,"position":11,"is_corresponding":false},{"id":29479,"name":"Ling Zhou","orcid":"0000-0002-5851-9492","position":12,"is_corresponding":false},{"id":73848,"name":"Zhijun Xiang","orcid":null,"position":13,"is_corresponding":false},{"id":113521,"name":"Jia-Ning Xiang","orcid":null,"position":14,"is_corresponding":false},{"id":113522,"name":"Stewart Leung","orcid":null,"position":15,"is_corresponding":false},{"id":113523,"name":"Liming Shao","orcid":"0000-0003-0694-7011","position":16,"is_corresponding":false},{"id":73850,"name":"Xichen Lin","orcid":null,"position":17,"is_corresponding":false},{"id":73845,"name":"Mercedes Lobera","orcid":"0000-0003-0803-1285","position":18,"is_corresponding":false},{"id":113524,"name":"Feng Ren","orcid":"0000-0001-9157-9182","position":19,"is_corresponding":false},{"id":73841,"name":"Yonghui Wang","orcid":"0000-0002-0262-2431","position":0,"is_corresponding":false}],"reference_count":0,"raw_metadata":{"has_enrichment":true,"base_score":3.4339872044851463,"endowment":3.4339872044851463,"datacite_reuse_total":0,"file_count":0,"downloads":0,"views":0,"has_version_chain":false,"is_dataset":false,"is_oa":false,"pmid":"29456799","pmcid":"PMC5807863","openalex_id":"https://openalex.org/W2784406062","authors":[],"funders":[{"funder_name":"National Natural Science Foundation of China","grant_id":"81573276","title":null},{"funder_name":"GlaxoSmithKline","grant_id":"","title":null}],"total_grants":2,"fwci":2.1293,"citation_percentile":0.87002252,"influential_citations":0,"citation_trend":[{"year":2018,"count":6},{"year":2019,"count":8},{"year":2020,"count":2},{"year":2021,"count":6},{"year":2022,"count":2},{"year":2023,"count":3},{"year":2025,"count":2},{"year":2026,"count":1}],"oa_status":"green","license":null,"oa_locations":[{"url":"https://www.ncbi.nlm.nih.gov/pmc/articles/5807863","host_type":"repository"},{"url":"https://europepmc.org/articles/pmc5807863?pdf=render","host_type":"GREEN"},{"url":"https://www.ncbi.nlm.nih.gov/pmc/articles/5807863","host_type":"repository"},{"url":"https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.7b00476","host_type":"publisher"},{"url":"https://doi.org/10.1021/acsmedchemlett.7b00476","host_type":"journal"},{"url":"https://pubmed.ncbi.nlm.nih.gov/29456799","host_type":"repository"},{"url":"http://europepmc.org/pmc/articles/PMC5807863","host_type":"repository"},{"url":"https://doi.org/10.7270/q2q81gm4","host_type":"repository"}],"fields_of_study":["Psoriasis: Treatment and Pathogenesis","NF-κB Signaling Pathways","Fungal Plant Pathogen Control","Medicine","Chemistry"],"mesh_terms":[],"keywords":["Inverse agonist","Agonist","RAR-related orphan receptor gamma","Corepressor","Coactivator","Amide","Chemistry","Orphan receptor","Peptide","Receptor","Nuclear receptor","Ligand (biochemistry)","Moiety","Computational biology","Stereochemistry","Biology","Biochemistry","Transcription factor","Gene"],"sdg_mappings":[{"sdg_number":0,"sdg_label":"Good health and well-being"}],"linked_datasets":[],"clinical_trials":[],"software_tools":[],"database_accessions":[{"name":"pdb"}],"source":"live","citation_network_status":"fetched"},"created_at":"2026-06-01T07:27:30.726124Z","pmid":null,"pmcid":null,"fwci":null,"citation_percentile":null,"influential_citations":0,"oa_status":null,"license":null,"views":0,"total_file_size_bytes":0,"version_count":0,"fair_f":null,"fair_a":null,"fair_i":null,"fair_r":null,"fair_zscore":null,"fair_rationale":null,"fair_model":null,"fair_agent_version":null,"fair_fulltext_source":null,"fair_has_llm":null,"fair_computed_at":null,"clinical_trials":[],"software_tools":[],"db_accessions":[],"linked_datasets":[],"topics":[]}