{"doi":"10.1016/j.ejmech.2022.114709","title":"Male contraceptive development: A medicinal chemistry perspective","abstract":"There is a need for non-hormonal contraceptives. One area that needs further investigation is the development of male contraceptives. Comparatively little is understood about potential drug targets in men to achieve a reversible contraceptive effect. In this article, we review the need for male contraceptives and some thoughts around the characteristics of a male contraceptive and the potential development pathway. We then discuss different potential approaches to discovering male contraceptives and then highlight potential targets that have been discussed in the literature.","journal":"European Journal of Medicinal Chemistry","year":2022,"id":273080,"datarank":0.0,"base_score":0.0,"endowment":0.0,"self_citation_contribution":0.0,"citation_network_contribution":0.0,"self_endowment_contribution":0.0,"citer_contribution":0.0,"corpus_percentile":null,"corpus_rank":null,"citation_count":11,"citer_count":0,"citers_with_citation_signal":0,"citers_with_endowment":0,"datacite_reuse_total":0,"is_dataset":false,"is_dataset_confidence":0.9555,"is_data_producer":false,"deposit_databanks":null,"is_oa":true,"file_count":0,"downloads":0,"has_version_chain":false,"published_date":"2022-01-01","fair_score":null,"fair_percentile":null,"algorithm_id":"datarank_citation_only_1hop_v6","ranking_scope":"data_only","authors":[{"id":940080,"name":"Irene Georgiou","orcid":"0000-0002-6042-9816","position":1,"is_corresponding":false},{"id":940081,"name":"Zoe C Johnston","orcid":"0000-0003-0904-7166","position":2,"is_corresponding":false},{"id":940082,"name":"Franz Gruber","orcid":"0000-0003-2008-8460","position":3,"is_corresponding":false},{"id":37917,"name":"Jason R. Swedlow","orcid":"0000-0002-2198-1958","position":4,"is_corresponding":false},{"id":592303,"name":"Kevin D. Read","orcid":"0000-0002-8536-0130","position":5,"is_corresponding":false},{"id":45011,"name":"Christopher L. R. Barratt","orcid":"0000-0003-0062-9979","position":6,"is_corresponding":false},{"id":587297,"name":"Ian H. Gilbert","orcid":"0000-0002-5238-1314","position":7,"is_corresponding":false},{"id":940079,"name":"Neil R. Norcross","orcid":"0000-0001-8050-5217","position":0,"is_corresponding":true}],"reference_count":101,"raw_metadata":null,"created_at":"2026-07-19T00:27:52.048702Z","pmid":"36087385","pmcid":null,"fwci":null,"citation_percentile":null,"influential_citations":0,"oa_status":null,"license":null,"views":0,"total_file_size_bytes":0,"version_count":0,"fair_f":null,"fair_a":null,"fair_i":null,"fair_r":null,"fair_zscore":null,"fair_rationale":null,"fair_model":null,"fair_agent_version":null,"fair_fulltext_source":null,"fair_has_llm":null,"fair_computed_at":null,"clinical_trials":[],"software_tools":[],"db_accessions":[],"linked_datasets":[],"topics":[]}