{"doi":"10.1016/j.bmcl.2020.127204","title":"Substituted benzyloxytricyclic compounds as retinoic acid-related orphan receptor gamma t (RORγt) agonists","abstract":null,"journal":"Bioorganic &amp; Medicinal Chemistry Letters","year":2020,"id":14473,"datarank":0.7871625413638237,"base_score":2.5649493574615367,"endowment":2.5649493574615367,"self_citation_contribution":0.38474240361923057,"citation_network_contribution":0.4024201377445931,"self_endowment_contribution":0.38474240361923057,"citer_contribution":0.4024201377445931,"corpus_percentile":null,"corpus_rank":null,"citation_count":12,"citer_count":11,"citers_with_citation_signal":11,"citers_with_endowment":11,"datacite_reuse_total":0,"is_dataset":false,"is_dataset_confidence":null,"is_oa":false,"file_count":0,"downloads":0,"has_version_chain":false,"published_date":null,"fair_score":null,"fair_percentile":null,"algorithm_id":"datarank_citation_only_1hop_v6","ranking_scope":"data_only","authors":[{"id":114173,"name":"Patrice Gill","orcid":null,"position":1,"is_corresponding":false},{"id":114174,"name":"Muthoni G. Kamau","orcid":null,"position":2,"is_corresponding":false},{"id":114175,"name":"Lan-Ying Qin","orcid":"0000-0003-2680-9986","position":3,"is_corresponding":false},{"id":112748,"name":"Zheming Ruan","orcid":null,"position":4,"is_corresponding":false},{"id":112753,"name":"Daniel O'Malley","orcid":null,"position":5,"is_corresponding":false},{"id":114176,"name":"Tram Huynh","orcid":null,"position":6,"is_corresponding":false},{"id":112754,"name":"Sylwia Stachura","orcid":null,"position":7,"is_corresponding":false},{"id":112756,"name":"Cullen L. Cavallaro","orcid":"0000-0001-9498-2612","position":8,"is_corresponding":false},{"id":114177,"name":"Zhonghui Lu","orcid":null,"position":9,"is_corresponding":false},{"id":114178,"name":"James J.-W. Duan","orcid":null,"position":10,"is_corresponding":false},{"id":112757,"name":"Carolyn A. Weigelt","orcid":null,"position":11,"is_corresponding":false},{"id":112758,"name":"John S. Sack","orcid":"0000-0003-1542-9515","position":12,"is_corresponding":false},{"id":112759,"name":"Max Ruzanov","orcid":null,"position":13,"is_corresponding":false},{"id":66995,"name":"Javed Khan","orcid":null,"position":14,"is_corresponding":false},{"id":112760,"name":"Murali Gururajan","orcid":null,"position":15,"is_corresponding":false},{"id":112761,"name":"Jessica J. Wong","orcid":null,"position":16,"is_corresponding":false},{"id":112762,"name":"Yanling Huang","orcid":null,"position":17,"is_corresponding":false},{"id":112763,"name":"Melissa Yarde","orcid":null,"position":18,"is_corresponding":false},{"id":112764,"name":"Zhuyin Li","orcid":null,"position":19,"is_corresponding":false},{"id":112765,"name":"Cliff Chen","orcid":null,"position":20,"is_corresponding":false},{"id":112766,"name":"Huadong Sun","orcid":null,"position":21,"is_corresponding":false},{"id":112767,"name":"Virna Borowski","orcid":null,"position":22,"is_corresponding":false},{"id":114179,"name":"Anwar Murtaza","orcid":null,"position":23,"is_corresponding":false},{"id":112771,"name":"Brian E. Fink","orcid":null,"position":24,"is_corresponding":false},{"id":112772,"name":"Lalgudi S. Harikrishnan","orcid":"0000-0002-4976-2933","position":0,"is_corresponding":false}],"reference_count":0,"raw_metadata":{"has_enrichment":true,"base_score":2.5649493574615367,"endowment":2.5649493574615367,"datacite_reuse_total":0,"file_count":0,"downloads":0,"views":0,"has_version_chain":false,"is_dataset":false,"is_oa":false,"pmid":"32334911","pmcid":null,"openalex_id":"https://openalex.org/W3019500503","authors":[],"funders":[],"total_grants":0,"fwci":0.9196,"citation_percentile":0.72841323,"influential_citations":0,"citation_trend":[{"year":2020,"count":1},{"year":2021,"count":5},{"year":2022,"count":2},{"year":2023,"count":3},{"year":2024,"count":1}],"oa_status":"green","license":"https://www.elsevier.com/legal/tdmrep-license","oa_locations":[{"url":"https://doi.org/10.7270/q2gx4g5t","host_type":"repository"},{"url":"https://doi.org/10.7270/q2gx4g5t","host_type":"repository"},{"url":"https://api.elsevier.com/content/article/PII:S0960894X20303048?httpAccept=text/xml","host_type":"publisher"},{"url":"https://api.elsevier.com/content/article/PII:S0960894X20303048?httpAccept=text/plain","host_type":"publisher"},{"url":"https://doi.org/10.1016/j.bmcl.2020.127204","host_type":"journal"},{"url":"https://pubmed.ncbi.nlm.nih.gov/32334911","host_type":"repository"}],"fields_of_study":["Retinoids in leukemia and cellular processes","Psoriasis: Treatment and Pathogenesis","Estrogen and related hormone effects","Chemistry","Medicine","Animals","Benzyl Compounds","Dose-Response Relationship, Drug","Female","Heterocyclic Compounds","Mice","Mice, Inbred C57BL","Molecular Structure","Receptors, Retinoic Acid","Structure-Activity Relationship","Retinoic Acid Receptor gamma"],"mesh_terms":["Retinoic Acid Receptor gamma","Animals","Benzyl Compounds","Dose-Response Relationship, Drug","Female","Heterocyclic Compounds","Mice, Inbred C57BL","Structure-Activity Relationship","Molecular Structure","Receptors, Retinoic Acid","Mice"],"keywords":["Chemistry","Orphan receptor","Agonist","Pharmacokinetics","Tricyclic","Retinoic acid","Pharmacodynamics","RAR-related orphan receptor gamma","Pharmacology","Stereochemistry","Chemical synthesis","Retinoic acid receptor","Receptor","In vitro","Biochemistry","Medicine","Rorγt","Rorgt","Ror Gamma","Retinoic Acid Related Orphan Receptor","Th17 Cells And Il-17"],"sdg_mappings":[{"sdg_number":0,"sdg_label":"Good health and well-being"}],"linked_datasets":[],"clinical_trials":[],"software_tools":[],"database_accessions":[],"source":"live","citation_network_status":"fetched"},"created_at":"2026-06-01T10:29:26.888390Z","pmid":null,"pmcid":null,"fwci":null,"citation_percentile":null,"influential_citations":0,"oa_status":null,"license":null,"views":0,"total_file_size_bytes":0,"version_count":0,"fair_f":null,"fair_a":null,"fair_i":null,"fair_r":null,"fair_zscore":null,"fair_rationale":null,"fair_model":null,"fair_agent_version":null,"fair_fulltext_source":null,"fair_has_llm":null,"fair_computed_at":null,"clinical_trials":[],"software_tools":[],"db_accessions":[],"linked_datasets":[],"topics":[]}