{"doi":"10.1016/j.bmc.2014.01.023","title":"Development of novel silicon-containing inverse agonists of retinoic acid receptor-related orphan receptors","abstract":null,"journal":"Bioorganic &amp; Medicinal Chemistry","year":2014,"id":14474,"datarank":1.3122707554966397,"base_score":2.995732273553991,"endowment":2.995732273553991,"self_citation_contribution":0.4493598410330987,"citation_network_contribution":0.8629109144635412,"self_endowment_contribution":0.4493598410330987,"citer_contribution":0.8629109144635412,"corpus_percentile":null,"corpus_rank":null,"citation_count":19,"citer_count":18,"citers_with_citation_signal":17,"citers_with_endowment":17,"datacite_reuse_total":1,"is_dataset":false,"is_dataset_confidence":null,"is_oa":false,"file_count":0,"downloads":0,"has_version_chain":false,"published_date":null,"fair_score":null,"fair_percentile":null,"algorithm_id":"datarank_citation_only_1hop_v6","ranking_scope":"data_only","authors":[{"id":114181,"name":"Masaharu Nakamura","orcid":null,"position":1,"is_corresponding":false},{"id":112619,"name":"Masahiko Nakamura","orcid":null,"position":2,"is_corresponding":false},{"id":114182,"name":"Yotaro Matsumoto","orcid":null,"position":3,"is_corresponding":false},{"id":112621,"name":"Madoka Nakagomi","orcid":null,"position":4,"is_corresponding":false},{"id":112624,"name":"Yuichi Hashimoto","orcid":null,"position":5,"is_corresponding":false},{"id":114180,"name":"Hirozumi Toyama","orcid":null,"position":0,"is_corresponding":false}],"reference_count":0,"raw_metadata":{"has_enrichment":true,"base_score":2.995732273553991,"endowment":2.995732273553991,"datacite_reuse_total":1,"file_count":0,"downloads":0,"views":0,"has_version_chain":false,"is_dataset":false,"is_oa":false,"pmid":"24559867","pmcid":null,"openalex_id":"https://openalex.org/W2037264551","authors":[],"funders":[],"total_grants":0,"fwci":1.5638,"citation_percentile":0.82344375,"influential_citations":0,"citation_trend":[{"year":2015,"count":3},{"year":2016,"count":3},{"year":2017,"count":5},{"year":2018,"count":2},{"year":2019,"count":1},{"year":2020,"count":1},{"year":2022,"count":1},{"year":2023,"count":1},{"year":2024,"count":2}],"oa_status":"green","license":"https://www.elsevier.com/legal/tdmrep-license","oa_locations":[{"url":"https://doi.org/10.7270/q25t3n0f","host_type":"repository"},{"url":"https://doi.org/10.7270/q25t3n0f","host_type":"repository"},{"url":"https://api.elsevier.com/content/article/PII:S0968089614000510?httpAccept=text/plain","host_type":"publisher"},{"url":"https://api.elsevier.com/content/article/PII:S0968089614000510?httpAccept=text/xml","host_type":"publisher"},{"url":"https://doi.org/10.1016/j.bmc.2014.01.023","host_type":"journal"},{"url":"https://pubmed.ncbi.nlm.nih.gov/24559867","host_type":"repository"}],"fields_of_study":["Retinoids in leukemia and cellular processes","Estrogen and related hormone effects","Nuclear Receptors and Signaling","Chemistry","Medicine","Anilides","Benzoates","Dose-Response Relationship, Drug","Drug Design","Humans","Models, Molecular","Molecular Structure","Nuclear Receptor Subfamily 1, Group F, Member 1","Organosilicon Compounds","Silicon","Structure-Activity Relationship","Tetrahydronaphthalenes"],"mesh_terms":["Anilides","Benzoates","Dose-Response Relationship, Drug","Humans","Models, Molecular","Silicon","Structure-Activity Relationship","Tetrahydronaphthalenes","Drug Design","Molecular Structure","Organosilicon Compounds","Nuclear Receptor Subfamily 1, Group F, Member 1"],"keywords":["Chemistry","Orphan receptor","Inverse agonist","Retinoic acid-inducible orphan G protein-coupled receptor","Retinoic acid","Receptor","Retinoic acid receptor","Retinoic acid receptor gamma","Biochemistry","Pharmacology","Stereochemistry","Agonist","Transcription factor","Gene","Silicon","Retinoic Acid Receptor-related Orphan Receptor"],"sdg_mappings":[{"sdg_number":0,"sdg_label":"Clean water and sanitation"}],"linked_datasets":[{"doi":"10.7270/q25t3n0f","title":"BindingDB Entry 50043915: Development of novel silicon-containing inverse agonists of retinoic acid receptor-related orphan receptors.","publisher":"BindingDB","resource_type":"Dataset"}],"clinical_trials":[],"software_tools":[],"database_accessions":[],"source":"live","citation_network_status":"fetched"},"created_at":"2026-06-01T10:30:09.034135Z","pmid":null,"pmcid":null,"fwci":null,"citation_percentile":null,"influential_citations":0,"oa_status":null,"license":null,"views":0,"total_file_size_bytes":0,"version_count":0,"fair_f":null,"fair_a":null,"fair_i":null,"fair_r":null,"fair_zscore":null,"fair_rationale":null,"fair_model":null,"fair_agent_version":null,"fair_fulltext_source":null,"fair_has_llm":null,"fair_computed_at":null,"clinical_trials":[],"software_tools":[],"db_accessions":[],"linked_datasets":[],"topics":[]}