{"doi":"10.1002/jlcr.3975","title":"Automated synthesis of <i>(R)</i>‐[<sup>18</sup>F]MH.MZ on the iPhase Flexlab reaction platform","abstract":"(R) ‐[ 18 F]MH.MZ ([ 18 F]MH.MZ) is a promising positron emission tomography (PET) radiotracer for in vivo study of the 5‐HT 2A receptor. To facilitate clinical trials, a fully automated radiosynthesis procedure for [ 18 F]MH.MZ was developed using commercially available materials on the iPhase Flexlab module. The overall synthesis time was 100 min with a radiochemical yield of 7 ± 0.9% ( n = 3). The radiochemical purity was greater than 99% for [ 18 F]MH.MZ with a molar activity of 361 ± 57 GBq/μmol ( n = 3). The protocol described herein reliably provides [ 18 F]MH.MZ that meets all relevant release criteria for a GMP radiopharmaceutical.","journal":"Journal of Labelled Compounds and Radiopharmaceuticals","year":2022,"id":294453,"datarank":0.16479184330021646,"base_score":1.0986122886681096,"endowment":1.0986122886681096,"self_citation_contribution":0.16479184330021646,"citation_network_contribution":0.0,"self_endowment_contribution":0.16479184330021646,"citer_contribution":0.0,"corpus_percentile":null,"corpus_rank":null,"citation_count":2,"citer_count":0,"citers_with_citation_signal":0,"citers_with_endowment":0,"datacite_reuse_total":0,"is_dataset":false,"is_dataset_confidence":0.9605,"is_data_producer":false,"deposit_databanks":null,"is_oa":true,"file_count":0,"downloads":0,"has_version_chain":false,"published_date":"2022-01-01","fair_score":null,"fair_percentile":null,"algorithm_id":"datarank_citation_only_1hop_v6","ranking_scope":"data_only","authors":[{"id":980180,"name":"Yiu‐Yin Cheung","orcid":null,"position":1,"is_corresponding":false},{"id":648391,"name":"Fei Liu","orcid":"0009-0005-0576-440X","position":2,"is_corresponding":false},{"id":698003,"name":"Todd E. Peterson","orcid":"0000-0002-5951-7384","position":3,"is_corresponding":false},{"id":888636,"name":"James F. Silverman","orcid":null,"position":4,"is_corresponding":false},{"id":883818,"name":"Ciaran Considine","orcid":"0000-0002-8171-2821","position":5,"is_corresponding":false},{"id":388676,"name":"Daniel O. Claassen","orcid":"0000-0002-9853-4902","position":6,"is_corresponding":false},{"id":775885,"name":"Adam J. Rosenberg","orcid":"0000-0003-2459-7043","position":0,"is_corresponding":true}],"reference_count":19,"raw_metadata":{"citation_network_status":"fetched"},"created_at":"2026-07-19T00:31:01.450041Z","pmid":"35491085","pmcid":null,"fwci":null,"citation_percentile":null,"influential_citations":0,"oa_status":null,"license":null,"views":0,"total_file_size_bytes":0,"version_count":0,"fair_f":null,"fair_a":null,"fair_i":null,"fair_r":null,"fair_zscore":null,"fair_rationale":null,"fair_model":null,"fair_agent_version":null,"fair_fulltext_source":null,"fair_has_llm":null,"fair_computed_at":null,"clinical_trials":[],"software_tools":[],"db_accessions":[],"linked_datasets":[],"topics":[]}